由1,2-胺醇制備氮雜環丙烷的反應。
羥基先和硫酸反應制備磺酸鹽，然后在堿作用下銨脫質子進行分子內親核取代關環得到產物：
An Improved and Mild Wenker Synthesis of Aziridines
X. Li, N. Chen, J. Xu, Synthesis, 2010, 3315-3318.
Synthesis of N-H vinylaziridines: a comparative study
B. Olofsson, R. Wijtmans, P. Somfai, Tetrahedron, 2002, 58, 5979-5982.
Short and Efficient Synthesis of Optically Active N-Tosyl Aziridines from 2-Amino Alcohols
L. W. Bieber, M. C. F. de Araujo, Molecules, 2002, 7, 902.
Generation and Ring Opening of Aziridines in Telescoped Continuous Flow Processes
N. Hsueh, G. J. Clarkson, M. Shipman, Org. Lett., 2015, 17, 3632-3635.
編譯自：Organic Chemistry Portal：http://www.organic-
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